LIST OF BINDING INTERFACES for query 'ALPHA-1' in category 'PROTEIN NAME'

(Click on the 'Details' column to view details on interfaces and similar patterns of amino acids)
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PDB Ligand Drug Indication Macromolecule/
Organism
Pfam Binding_Interfaces (View) Details
3apv TP0Amitriptyline
(DB00321)
Amitriptyline is a tricyclic antidepressant indicated in the treatment of depressive illness, either endogenous or psychotic, and to relieve depression associated anxiety.ALPHA-1-ACID GLYCOPROTEIN 2
(Homo sapiens)
Lipocalin
3apw DP0Disopyramide
(DB00280)
Disopyramide is a class 1A antiarrhythmic agent used to treat life-threatening ventricular arrhythmias.ALPHA-1-ACID GLYCOPROTEIN 2
(Homo sapiens)
Lipocalin
3apx Z80Chlorpromazine
(DB00477)
Chlorpromazine is a phenothiazine antipsychotic used to treat nausea, vomiting, preoperative anxiety, schizophrenia, bipolar disorder, and severe behavioral problems in children.ALPHA-1-ACID GLYCOPROTEIN 2
(Homo sapiens)
Lipocalin
5j2t VLBVinblastine
(DB00570)
Vinblastine is a vinca alkaloid used to treat breast cancer, testicular cancer, neuroblastoma, Hodgkin's and non-Hodgkins lymphoma, mycosis fungoides, histiocytosis, and Kaposi's sarcoma.TUBULIN ALPHA-1B CHAIN;
TUBULIN BETA-2B CHAIN
(Rattus norvegicus;
gallus gallus;
bos taurus
)
Tubulin
Tubulin_C
5jh7 6K9Eribulin
(DB08871)
Eribulin is a microtubule inhibitor used to treat metastatic breast cancer and metastatic or unresectable liposarcoma.TUBULIN ALPHA-1B CHAIN;
TUBULIN BETA-2B CHAIN
(Rattus norvegicus;
gallus gallus;
bos taurus
)
Tubulin
Tubulin_C
5om2 DXTDoxycycline
(DB00254)
Doxycycline is a tetracycline antibiotic used to treat a wide variety of bacterial infections.ALPHA-1-ANTICHYMOTRYPSIN
(Homo sapiens)
NA
5om7 DM2Doxorubicin
(DB00997)
Doxorubicin is a medication used to treat various cancers and Kaposi's Sarcoma.ALPHA-1-ANTICHYMOTRYPSIN
(Homo sapiens)
NA
6dw0 ABUGamma-aminobutyric acid
(DB02530)
The most common inhibitory neurotransmitter in the central nervous system.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-1
(Rattus norvegicus)
Neur_chan_LBD
Neur_chan_memb
6dw1 ABUGamma-aminobutyric acid
(DB02530)
The most common inhibitory neurotransmitter in the central nervous system.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-1
(Rattus norvegicus)
Neur_chan_LBD
Neur_chan_memb
6ftp DM2Doxorubicin
(DB00997)
Doxorubicin is a medication used to treat various cancers and Kaposi's Sarcoma.ALPHA-1-ANTICHYMOTRYPSIN
(Homo sapiens)
NA
6hgf HCYHydrocortisone
(DB00741)
Hydrocortisone is a glucocorticoid used to treat corticosteroid-responsive dermatoses, endocrine disorders, immune conditions, and allergic disorders.ALPHA-1-ANTICHYMOTRYPSIN
(Homo sapiens)
NA
6hgg HCYHydrocortisone
(DB00741)
Hydrocortisone is a glucocorticoid used to treat corticosteroid-responsive dermatoses, endocrine disorders, immune conditions, and allergic disorders.ALPHA-1-ANTICHYMOTRYPSIN
(Homo sapiens)
NA
6hgk STRProgesterone
(DB00396)
Progesterone is a hormone used for a variety of functions, including contraception, control of abnormal uterine bleeding, maintenance of pregnancy, and prevention of endometrial hyperplasia.ALPHA-1-ANTICHYMOTRYPSIN
(Homo sapiens)
NA
6hgl TESTestosterone
(DB00624)
Testosterone is a hormone used to treat hypogonadism, breast carcinoma in women, or the vasomotor symptoms of menopause.ALPHA-1-ANTICHYMOTRYPSIN
(Homo sapiens)
NA
6huj ABUGamma-aminobutyric acid
(DB02530)
The most common inhibitory neurotransmitter in the central nervous system.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-3
(Bos taurus;
homo sapiens;
lama glama
)
Neur_chan_LBD
Neur_chan_memb
6huo 08HAlprazolam
(DB00404)
Alprazolam is a triazolobenzodiazepine with intermediate onset commonly used to treat panic disorders and generalized anxiety in addition to anxiety associated with depression.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT GAMMA-2
(Bos taurus;
homo sapiens;
lama glama
)
Neur_chan_LBD
Neur_chan_memb
6huo ABUGamma-aminobutyric acid
(DB02530)
The most common inhibitory neurotransmitter in the central nervous system.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-3
(Bos taurus;
homo sapiens;
lama glama
)
Neur_chan_LBD
Neur_chan_memb
6hup DZPDiazepam
(DB00829)
Diazepam is a long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-3
(Bos taurus;
homo sapiens;
lama glama
)
Neur_chan_LBD
Neur_chan_memb
6hup DZPDiazepam
(DB00829)
Diazepam is a long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT GAMMA-2
(Bos taurus;
homo sapiens;
lama glama
)
Neur_chan_LBD
Neur_chan_memb
6jp5 C5UNifedipine
(DB01115)
Nifedipine is a dihydropyridine calcium channel blocker indicated for the management of several subtypes of angina pectoris, and hypertension.VOLTAGE-DEPENDENT L-TYPE CALCIUM CHANNEL SUBUNIT ALPHA-1S
(Oryctolagus cuniculus)
CAC1F_C
Ca_chan_IQ
GPHH
Ion_trans
6jpb C9FDiltiazem
(DB00343)
Diltiazem is a calcium channel blocker used to treat hypertension and to manage chronic stable angina.VOLTAGE-DEPENDENT L-TYPE CALCIUM CHANNEL SUBUNIT ALPHA-1S
(Oryctolagus cuniculus)
CAC1F_C
Ca_chan_IQ
GPHH
Ion_trans
6x3t ABUGamma-aminobutyric acid
(DB02530)
The most common inhibitory neurotransmitter in the central nervous system.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
Neur_chan_memb
6x3u FYPFlumazenil
(DB01205)
Flumazenil is a benzodiazepine antagonist that is used for the complete or partial reversal of the sedative effects caused by benzodiazepines in various clinical settings, such as induced general anesthesia for diagnostic and therapeutic procedures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT GAMMA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
6x3v V8DEtomidate
(DB00292)
Etomidate is a short-acting intravenous anesthetic indicated for the induction of anesthesia and supplementation of subpotent anesthesia during short operative procedures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
Neur_chan_memb
6x3w UQAPhenobarbital
(DB01174)
Phenobarbital is a long-lasting barbiturate and anticonvulsant used in the treatment of all types of seizures, except for absent seizures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
Neur_chan_memb
6x3x DZPDiazepam
(DB00829)
Diazepam is a long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
Neur_chan_memb
6x3x DZPDiazepam
(DB00829)
Diazepam is a long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT GAMMA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
7ddh DGXDigoxin
(DB00390)
Digoxin is a cardiac glycoside used in the treatment of mild to moderate heart failure and for ventricular response rate control in chronic atrial fibrillation.SODIUM/POTASSIUM-TRANSPORTING ATPASE SUBUNIT ALPHA-1;
SODIUM/POTASSIUM-TRANSPORTING ATPASE SUBUNIT BETA-1
(Sus scrofa)
Cation_ATPase
Cation_ATPase_C
Cation_ATPase_N
E1-E2_ATPase
Na_K-ATPase
7ddi F9RDigitoxin
(DB01396)
Digitoxin is a cardiac glycoside used in the treatment and management of congestive cardiac insufficiency, arrhythmias and heart failure.SODIUM/POTASSIUM-TRANSPORTING ATPASE SUBUNIT ALPHA-1;
SODIUM/POTASSIUM-TRANSPORTING ATPASE SUBUNIT BETA-1
(Sus scrofa)
Cation_ATPase
Cation_ATPase_C
Cation_ATPase_N
E1-E2_ATPase
Na_K-ATPase
7ddj OBNOuabain
(DB01092)
A cardioactive glycoside consisting of rhamnose and ouabagenin, obtained from the seeds of Strophanthus gratus and other plants of the Apocynaceae; used like digitalis. It is commonly used in cell...SODIUM/POTASSIUM-TRANSPORTING ATPASE SUBUNIT ALPHA-1
(Sus scrofa)
Cation_ATPase
Cation_ATPase_C
Cation_ATPase_N
E1-E2_ATPase
7jpx 6UBLevamlodipine
(DB09237)
Levamlodipine is a calcium channel blocker used to treat hypertension.VOLTAGE-DEPENDENT L-TYPE CALCIUM CHANNEL SUBUNIT ALPHA-1S
(Oryctolagus cuniculus)
CAC1F_C
Ca_chan_IQ
GPHH
Ion_trans
PDB Ligand Drug Indication Macromolecule/
Organism
Pfam Binding_Interfaces (View) Details