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| PDB | Ligand | Drug | Indication | Macromolecule/ Organism |
Pfam | Binding_Interfaces (View) | Details |
|---|---|---|---|---|---|---|---|
| 1l2i | CCS | Carbocisteine (DB04339) | Carbocisteine is a expectorant mucolytic used in the relief of respiratory of COPD and other conditions associated with increased mucus viscosity. | ESTROGEN RECEPTOR (Homo sapiens;synthetic construct) | Hormone_recep | ||
| 1qkn | RAL | Raloxifene (DB00481) | Raloxifene is a selective estrogen receptor modulator that is used to prevent and treat osteoporosis and reduce the risk of invasive breast cancer in high-risk postmenopausal women. | ESTROGEN RECEPTOR BETA (Rattus norvegicus) | Hormone_recep | ||
| 2qxs | RAL | Raloxifene (DB00481) | Raloxifene is a selective estrogen receptor modulator that is used to prevent and treat osteoporosis and reduce the risk of invasive breast cancer in high-risk postmenopausal women. | ESTROGEN RECEPTOR (Homo sapiens) | Hormone_recep | ||
| 3hm1 | J3Z | Estrone (DB00655) | Estrone is an estrogen used to treat perimenopausal and postmenopausal symptoms. | ESTROGEN RECEPTOR (Homo sapiens;synthetic construct) | Hormone_recep | ||
| 3oll | EST | Estradiol (DB00783) | Estradiol is an estrogenic steroid used to treat vasomotor symptoms of vulvar and vaginal atrophy in menopause, hypoestrogenism, prevention of postmenopausal osteoporosis, treatment of breast cancer, and advanced androgen-dependent carcinoma of the prostate. | ESTROGEN RECEPTOR BETA (Homo sapiens;synthetic construct) | Hormone_recep | ||
| 3q95 | ESL | Estriol (DB04573) | Estriol is a weak estrogen used to treat vaginal dryness and estrogen deficiency conditions, such as vaginitis and vulvar itching. | ESTROGEN RECEPTOR (Homo sapiens;synthetic construct) | Hormone_recep | ||
| 4mg8 | 27J | Zeranol (DB11478) | Zeranol is a non-steroidal estrogen agonist. It is a mycotoxin, derived from fungi in the Fusarium family, and may be found as a contaminant in fungus-infected crops. It is 3-4x... | ESTROGEN RECEPTOR (Homo sapiens;synthetic construct) | Hormone_recep | ||
| 4tv1 | 36M | Propylparaben (DB14177) | Propylparaben is used in allergenic testing. | ESTROGEN RECEPTOR (Homo sapiens;synthetic construct) | Hormone_recep | ||
| 4zn7 | DES | Diethylstilbestrol (DB00255) | A synthetic nonsteroidal estrogen used in the treatment of menopausal and postmenopausal disorders. It was also used formerly as a growth promoter in animals. According to the Fourth Annual Report... | ESTROGEN RECEPTOR (Homo sapiens;synthetic construct) | Hormone_recep | ||
| 5dxe | EST | Estradiol (DB00783) | Estradiol is an estrogenic steroid used to treat vasomotor symptoms of vulvar and vaginal atrophy in menopause, hypoestrogenism, prevention of postmenopausal osteoporosis, treatment of breast cancer, and advanced androgen-dependent carcinoma of the prostate. | ESTROGEN RECEPTOR (Homo sapiens;synthetic construct) | Hormone_recep | ||
| 6psj | 29S | Bazedoxifene (DB06401) | Bazedoxifene is a selective estrogen receptor modulator (SERM) used to treat moderate to severe vasomotor symptoms in menopause and osteoporosis alone or in combination with conjugated estrogens. | ESTROGEN RECEPTOR (Homo sapiens) | Hormone_recep | ||
| 6vjd | C3D | Lasofoxifene (DB06202) | Lasofoxifene is a non-steroidal 3rd generation selective estrogen receptor modulator (SERM) that selectively binds to both ERα and ERβ with high affinity. It is a naphthalene derivative marketed for prevention... | ESTROGEN RECEPTOR (Homo sapiens) | Hormone_recep | ||
| PDB | Ligand | Drug | Indication | Macromolecule/ Organism |
Pfam | Binding_Interfaces (View) | Details |