LIST OF BINDING INTERFACES for query 'GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1' in category 'PROTEIN NAME'

(Click on the 'Details' column to view details on interfaces and similar patterns of amino acids)
Click on the 'View' column to view patterns on the structural viewer)
PDB Ligand Drug Indication Macromolecule/
Organism
Pfam Binding_Interfaces (View) Details
6dw0 ABUGamma-aminobutyric acid
(DB02530)
The most common inhibitory neurotransmitter in the central nervous system.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-1
(Rattus norvegicus)
Neur_chan_LBD
Neur_chan_memb
6dw1 ABUGamma-aminobutyric acid
(DB02530)
The most common inhibitory neurotransmitter in the central nervous system.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-1
(Rattus norvegicus)
Neur_chan_LBD
Neur_chan_memb
6huj ABUGamma-aminobutyric acid
(DB02530)
The most common inhibitory neurotransmitter in the central nervous system.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-3
(Bos taurus;
homo sapiens;
lama glama
)
Neur_chan_LBD
Neur_chan_memb
6huo 08HAlprazolam
(DB00404)
Alprazolam is a triazolobenzodiazepine with intermediate onset commonly used to treat panic disorders and generalized anxiety in addition to anxiety associated with depression.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT GAMMA-2
(Bos taurus;
homo sapiens;
lama glama
)
Neur_chan_LBD
Neur_chan_memb
6huo ABUGamma-aminobutyric acid
(DB02530)
The most common inhibitory neurotransmitter in the central nervous system.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-3
(Bos taurus;
homo sapiens;
lama glama
)
Neur_chan_LBD
Neur_chan_memb
6hup DZPDiazepam
(DB00829)
Diazepam is a long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-3
(Bos taurus;
homo sapiens;
lama glama
)
Neur_chan_LBD
Neur_chan_memb
6hup DZPDiazepam
(DB00829)
Diazepam is a long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1,GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT GAMMA-2
(Bos taurus;
homo sapiens;
lama glama
)
Neur_chan_LBD
Neur_chan_memb
6x3t ABUGamma-aminobutyric acid
(DB02530)
The most common inhibitory neurotransmitter in the central nervous system.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
Neur_chan_memb
6x3u FYPFlumazenil
(DB01205)
Flumazenil is a benzodiazepine antagonist that is used for the complete or partial reversal of the sedative effects caused by benzodiazepines in various clinical settings, such as induced general anesthesia for diagnostic and therapeutic procedures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT GAMMA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
6x3v V8DEtomidate
(DB00292)
Etomidate is a short-acting intravenous anesthetic indicated for the induction of anesthesia and supplementation of subpotent anesthesia during short operative procedures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
Neur_chan_memb
6x3w UQAPhenobarbital
(DB01174)
Phenobarbital is a long-lasting barbiturate and anticonvulsant used in the treatment of all types of seizures, except for absent seizures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
Neur_chan_memb
6x3x DZPDiazepam
(DB00829)
Diazepam is a long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT BETA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
Neur_chan_memb
6x3x DZPDiazepam
(DB00829)
Diazepam is a long-acting benzodiazepine with rapid onset commonly used to treat panic disorders, severe anxiety, alcohol withdrawal, and seizures.GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT GAMMA-2
(Homo sapiens;
mus musculus
)
Neur_chan_LBD
PDB Ligand Drug Indication Macromolecule/
Organism
Pfam Binding_Interfaces (View) Details