DRUG BINDING INTERFACES MAPPED TO 'GAMMA-AMINOBUTYRIC ACID RECEPTOR SUBUNIT GAMMA-2'

List of Binding Interfaces
(Click on the entry ID to view details of interfaces and pattern clusters)
(Note that ASSAM search use only 3-12 residue containing patterns)
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DrReposER ID PDB Ligand Organism Macromolecule Pfam Res. Interface HETATM
6D6U_D_FYPD410 6d6u FYP

DB01205
(Flumazenil)
Homo sapiens GAMMA-AMINOBUTYRIC
ACID RECEPTOR
SUBUNIT
ALPHA-1,GAMMA-AMINOB
UTYRIC ACID RECEPTOR
SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC
ACID RECEPTOR
SUBUNIT
GAMMA-2,GAMMA-AMINOB
UTYRIC ACID RECEPTOR
SUBUNIT GAMMA-2
None
PF02931
(Neur_chan_LBD)
PF02932
(Neur_chan_memb)
9 ASP E  56
TYR E  58
ALA E  79
HIS D 102
THR E 142
TYR D 160
SER D 205
SER D 206
TYR D 210
FYP D 410
6HUO_D_08HD501 6huo 08H

DB00404
(Alprazolam)
Homo sapiens;
Homo sapiens;
Bos taurus
GAMMA-AMINOBUTYRIC
ACID RECEPTOR
SUBUNIT
ALPHA-1,GAMMA-AMINOB
UTYRIC ACID RECEPTOR
SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC
ACID RECEPTOR
SUBUNIT GAMMA-2
None
PF02931
(Neur_chan_LBD)
PF02932
(Neur_chan_memb)
8 TYR C  58
ASN C  60
PHE C  77
PHE D 100
HIS D 102
VAL D 203
SER D 205
TYR D 210
08H D 501
6HUP_D_DZPD2001 6hup DZP

DB00829
(Diazepam)
Homo sapiens;
Homo sapiens;
Bos taurus
GAMMA-AMINOBUTYRIC
ACID RECEPTOR
SUBUNIT
ALPHA-1,GAMMA-AMINOB
UTYRIC ACID RECEPTOR
SUBUNIT ALPHA-1;
GAMMA-AMINOBUTYRIC
ACID RECEPTOR
SUBUNIT GAMMA-2
None
PF02931
(Neur_chan_memb)
PF02932
(Neur_chan_LBD)
9 TYR C  58
ASN C  60
PHE C  77
PHE D 100
HIS D 102
TYR D 160
VAL D 203
SER D 205
TYR D 210
DZP D2001