DRUG BINDING INTERFACES MAPPED TO 'DNA TOPOISOMERASE I'

List of Binding Interfaces
(Click on the entry ID to view details of interfaces and pattern clusters)
(Note that ASSAM search use only 3-12 residue containing patterns)
Filter list by:
DrReposER ID PDB Ligand Organism Macromolecule Pfam Res. Interface HETATM
1K4T_D_TTCD990 1k4t TTC

DB01030
(Topotecan)
;
Homo sapiens
DNA TOPOISOMERASE I PF01028
(Topoisom_I)
PF02919
(Topoisom_I_N)
PF14370
(Topo_C_assoc)
no annotation
5 GLU A 356
ARG A 364
LYS A 532
ASP A 533
THR A 718
TTC D 990
1QZR_B_CDXB901 1qzr CDX

DB00380
(Dexrazoxane)
Saccharomyces
cerevisiae
DNA TOPOISOMERASE II PF00204
(DNA_gyraseB)
PF02518
(HATPase_c)
no annotation
14 HIS A  20
HIS B  20
THR B  27
THR A  27
TYR A  28
TYR B  28
ASN B 142
ASN A 142
TYR B 144
TYR A 144
LEU A 148
LEU B 148
GLN B 365
GLN A 365
CDX B 901
1RR8_A_TTCA100 1rr8 TTC

DB01030
(Topotecan)
;
Homo sapiens
DNA TOPOISOMERASE I PF01028
(Topoisom_I)
PF02919
(Topoisom_I_N)
PF14370
(Topo_C_assoc)
no annotation
5 GLU C 356
ARG C 364
LYS C 532
ASP C 533
THR C 718
TTC A 100
1RRJ_B_TTCB990 1rrj TTC

DB01030
(Topotecan)
;
Homo sapiens
DNA TOPOISOMERASE I PF01028
(Topoisom_I)
PF02919
(Topoisom_I_N)
PF14370
(Topo_C_assoc)
no annotation
5 GLU A 356
ARG A 364
LYS A 532
ASP A 533
THR A 718
TTC B 990
4URN_A_NOVA2000 4urn NOV

DB01051
(Novobiocin)
Staphylococcus
aureus
DNA TOPOISOMERASE
IV, B SUBUNIT
PF02518
(HATPase_c)
no annotation
14 ASP B  35
LYS B  36
ASN A  49
SER A  50
ASP A  52
GLU A  53
ASP A  76
ARG A  79
MET A  81
PRO A  82
ILE A  96
ARG A 138
THR A 168
ASN B 186
NOV A2000
4URN_B_NOVB2000 4urn NOV

DB01051
(Novobiocin)
Staphylococcus
aureus
DNA TOPOISOMERASE
IV, B SUBUNIT
no annotation 11 ASN B  49
SER B  50
ASP B  52
GLU B  53
ASP B  76
ARG B  79
MET B  81
PRO B  82
ILE B  96
ARG B 138
THR B 168
NOV B2000
4URN_C_NOVC2000 4urn NOV

DB01051
(Novobiocin)
Staphylococcus
aureus
DNA TOPOISOMERASE
IV, B SUBUNIT
no annotation 11 ASN C  49
SER C  50
ASP C  52
GLU C  53
ASP C  76
ARG C  79
MET C  81
PRO C  82
ILE C  96
ARG C 138
THR C 168
NOV C2000