Ligand ID: LF7 Drugbank ID: DB04876(Vildagliptin) Indication:Used to reduce hyperglycemia in type 2 diabetes mellitus. |
DrReposER ID / Desc. | Hit PDBID |
Hit Macromolecule |
Res. Matches |
View | Interface | RMSD | Seq. Identity (%) |
HETATM | Dock | |
---|---|---|---|---|---|---|---|---|---|---|
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 1uk4 | 3C-LIKE PROTEINASE (SARSr-CoV) | 5 / 11 | ARG B 298TYR A 118VAL A 114TYR A 126VAL A 125 | 1.77A | 16.29 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 1uk4 | 3C-LIKE PROTEINASE (SARSr-CoV) | 5 / 12 | ARG B 298TYR A 118VAL A 114TYR A 126VAL A 125 | 1.75A | 16.19 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 1x7q | HLA, A-11 (Homosapiens) | 5 / 12 | ARG A 163TYR A 59TYR A 7ASN A 66VAL A 67 | 1.78A | 18.10 | SO4 A4003 (-4.0A)NoneNoneNoneNone | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 1x7q | HLA, A-11 (Homosapiens) | 5 / 12 | ARG A 163TYR A 59TYR A 7ASN A 66VAL A 67 | 1.78A | 18.09 | SO4 A4003 (-4.0A)NoneNoneNoneNone | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 1z1j | 3C-LIKE PROTEINASE (SARSr-CoV) | 5 / 12 | ARG A 298TYR B1118VAL B1114TYR B1126VAL B1125 | 1.78A | 16.29 | None | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 1z1j | 3C-LIKE PROTEINASE (SARSr-CoV) | 5 / 11 | ARG A 298TYR B1118VAL B1114TYR B1126VAL B1125 | 1.79A | 16.29 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 1z1j | 3C-LIKE PROTEINASE (SARSr-CoV) | 5 / 12 | ARG A 298TYR B1118VAL B1114TYR B1126VAL B1125 | 1.79A | 16.19 | None | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 2amq | 3C-LIKE PROTEINASE (SARSr-CoV) | 5 / 11 | ARG B 298TYR A 118VAL A 114TYR A 126VAL A 125 | 1.78A | 16.19 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 2amq | 3C-LIKE PROTEINASE (SARSr-CoV) | 5 / 12 | ARG B 298TYR A 118VAL A 114TYR A 126VAL A 125 | 1.76A | 16.19 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 2duc | REPLICASEPOLYPROTEIN 1AB (SARSr-CoV) | 5 / 12 | ARG B 298TYR A 118VAL A 114TYR A 126VAL A 125 | 1.75A | 16.29 | None | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 2fe8 | REPLICASEPOLYPROTEIN 1AB (SARSr-CoV) | 5 / 11 | ARG C 285GLU C 264SER C 116VAL C 166TYR C 265 | 1.66A | 17.61 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 2fe8 | REPLICASEPOLYPROTEIN 1AB (SARSr-CoV) | 5 / 12 | ARG C 285GLU C 264SER C 116VAL C 166TYR C 265 | 1.65A | 17.33 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 2fe8 | REPLICASEPOLYPROTEIN 1AB (SARSr-CoV) | 5 / 12 | ARG C 285GLU C 264SER C 116VAL C 166TYR C 265 | 1.66A | 17.61 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 3aw1 | 3C-LIKE PROTEINASE (SARSr-CoV) | 5 / 12 | ARG B 298TYR A 118VAL A 114TYR A 126VAL A 125 | 1.76A | 16.19 | None | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 3aw1 | 3C-LIKE PROTEINASE (SARSr-CoV) | 5 / 11 | ARG B 298TYR A 118VAL A 114TYR A 126VAL A 125 | 1.77A | 16.29 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 3aw1 | 3C-LIKE PROTEINASE (SARSr-CoV) | 5 / 12 | ARG B 298TYR A 118VAL A 114TYR A 126VAL A 125 | 1.76A | 16.29 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 3e9s | NSP3 (SARSr-CoV) | 5 / 12 | ARG A 285GLU A 264SER A 116VAL A 166TYR A 265 | 1.79A | 17.45 | NoneNoneOCS A 112 ( 3.7A)NoneTTT A 317 (-4.1A) | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 3to2 | MHC CLASS I ANTIGEN (Homosapiens) | 5 / 12 | TYR A 85TYR A 84TYR A 116TYR A 123VAL A 95 | 1.74A | 18.15 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 3to2 | MHC CLASS I ANTIGEN (Homosapiens) | 5 / 12 | TYR A 85TYR A 84TYR A 116TYR A 123VAL A 95 | 1.74A | 18.14 | None | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 3to2 | MHC CLASS I ANTIGEN (Homosapiens) | 5 / 11 | TYR A 85TYR A 84TYR A 116TYR A 123VAL A 95 | 1.75A | 18.15 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 5e6j | REPLICASEPOLYPROTEIN 1AB (SARSr-CoV) | 5 / 12 | GLU D 239TYR D 214TYR D 311VAL D 236VAL D 185 | 1.69A | 17.61 | None | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 5e6j | REPLICASEPOLYPROTEIN 1AB (SARSr-CoV) | 5 / 11 | GLU D 239TYR D 214TYR D 311VAL D 236VAL D 185 | 1.68A | 17.61 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 5e6j | REPLICASEPOLYPROTEIN 1AB (SARSr-CoV) | 5 / 12 | GLU D 239TYR D 214TYR D 311VAL D 236VAL D 185 | 1.68A | 18.11 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 5tl6 | REPLICASEPOLYPROTEIN 1AB (SARSr-CoV) | 5 / 12 | ARG D 139GLU D 135TYR D 84VAL D 12TYR D 72 | 1.66A | 17.31 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 5x5c | S PROTEIN (MERS-CoV) | 5 / 12 | GLU B 513TYR C 409VAL C 575TYR C 577ASN C 582 | 1.64A | 21.61 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 6crw | SPIKEGLYCOPROTEIN,FIBRITIN (SARSr-CoV) | 5 / 12 | ARG B 183GLU B 93VAL B 140ASN B 96VAL B 172 | 1.75A | 21.18 | None | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6crw | SPIKEGLYCOPROTEIN,FIBRITIN (SARSr-CoV) | 5 / 11 | ARG B 183GLU B 93VAL B 140ASN B 96VAL B 172 | 1.74A | 21.18 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6crw | SPIKEGLYCOPROTEIN,FIBRITIN (SARSr-CoV) | 5 / 12 | ARG B 183GLU B 93VAL B 140ASN B 96VAL B 172 | 1.75A | 21.20 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6m2n | 3CL PROTEASE (SARS-CoV-2) | 5 / 12 | ARG D 298TYR B 118VAL B 114TYR B 126VAL B 125 | 1.79A | 15.91 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6y2g | REPLICASEPOLYPROTEIN 1AB (SARS-CoV-2) | 5 / 12 | ARG A 298TYR B 118VAL B 114TYR B 126VAL B 125 | 1.80A | 15.91 | None | ||
![]() | 3W2T_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 6yla | LIGHT CHAIN (Homosapiens) | 5 / 12 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.76A | 15.89 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 6yla | LIGHT CHAIN (Homosapiens) | 5 / 12 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.78A | 18.41 | None | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6yla | LIGHT CHAIN (Homosapiens) | 5 / 11 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.77A | 18.41 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 6yla | LIGHT CHAIN (Homosapiens) | 5 / 12 | TYR C 102SER C 99TYR C 97VAL C 29TYR C 31 | 1.78A | 18.41 | NoneDMS C 303 (-4.1A)NoneNoneNone | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6yla | LIGHT CHAIN (Homosapiens) | 5 / 11 | TYR C 102SER C 99TYR C 97VAL C 29TYR C 31 | 1.77A | 18.41 | NoneDMS C 303 (-4.1A)NoneNoneNone | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6yla | LIGHT CHAIN (Homosapiens) | 5 / 12 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.75A | 15.89 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6yla | LIGHT CHAIN (Homosapiens) | 5 / 12 | TYR C 102SER C 99TYR C 97VAL C 29TYR C 31 | 1.75A | 15.89 | NoneDMS C 303 (-4.1A)NoneNoneNone | ||
![]() | 3W2T_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 6yla | LIGHT CHAIN (Homosapiens) | 5 / 12 | TYR C 102SER C 99TYR C 97VAL C 29TYR C 31 | 1.75A | 15.89 | NoneDMS C 303 (-4.1A)NoneNoneNone | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6ym0 | LIGHT CHAIN (Homosapiens) | 5 / 11 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.74A | 18.41 | None | ||
![]() | 3W2T_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 6ym0 | LIGHT CHAIN (Homosapiens) | 5 / 12 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.73A | 15.89 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 6ym0 | LIGHT CHAIN (Homosapiens) | 5 / 12 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.75A | 18.41 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6ym0 | LIGHT CHAIN (Homosapiens) | 5 / 12 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.72A | 15.89 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 6yor | IGG L CHAIN (Homosapiens) | 5 / 12 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.77A | 18.41 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6yor | IGG L CHAIN (Homosapiens) | 5 / 12 | TYR C 102SER C 99TYR C 97VAL C 29TYR C 31 | 1.75A | 15.89 | None | ||
![]() | 3W2T_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 6yor | IGG L CHAIN (Homosapiens) | 5 / 12 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.75A | 15.89 | None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6yor | IGG L CHAIN (Homosapiens) | 5 / 12 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.74A | 15.89 | None | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6yor | IGG L CHAIN (Homosapiens) | 5 / 11 | TYR L 102SER L 99TYR L 97VAL L 29TYR L 31 | 1.77A | 18.41 | None | ||
![]() | 3W2T_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 6yor | IGG L CHAIN (Homosapiens) | 5 / 12 | TYR C 102SER C 99TYR C 97VAL C 29TYR C 31 | 1.76A | 15.89 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 6yor | IGG L CHAIN (Homosapiens) | 5 / 12 | TYR C 102SER C 99TYR C 97VAL C 29TYR C 31 | 1.78A | 18.41 | None | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 6yor | IGG L CHAIN (Homosapiens) | 5 / 11 | TYR C 102SER C 99TYR C 97VAL C 29TYR C 31 | 1.77A | 18.41 | None | ||
![]() | 6B1E_B_LF7B801_1 (DIPEPTIDYL PEPTIDASE4) | 7bv2 | NSP12 (SARS-CoV-2) | 5 / 12 | ARG A 654GLU A 658SER A 564VAL A 560ASN A 568 | 1.34A | 20.04 | NoneNoneNone U T 10 ( 4.6A)None | ||
![]() | 6B1E_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 7bv2 | NSP12 (SARS-CoV-2) | 5 / 11 | ARG A 654GLU A 658SER A 564VAL A 560ASN A 568 | 1.33A | 20.04 | NoneNoneNone U T 10 ( 4.6A)None | ||
![]() | 3W2T_A_LF7A801_1 (DIPEPTIDYL PEPTIDASE4) | 7bv2 | NSP12 (SARS-CoV-2) | 5 / 12 | ARG A 654GLU A 658SER A 564VAL A 560ASN A 568 | 1.36A | 20.56 | NoneNoneNone U T 10 ( 4.6A)None |