POTENTIAL TARGETS FROM HUMAN (RESULTS FROM SUB-STRUCTURAL SIMILARITY SEARCHES)
1) User may click on the DrReposER ID (the second column) to get information on the binding sites and drug molecule.
2) Click View (the second last column) to view matched residues and superposition in the NGL viewer (upper right part).
3) User may also click on the Dock (the last column) to get script for molecular docking in UCSF Chimera through AutoDock Vina.


DrReposER ID / Desc. Hit
PDBID
Hit
Macromolecule
Res.
Matches
Interface HETATM RMSD Seq.
Identity (%)
View Dock
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
1kcw CERULOPLASMIN
(Homo
sapiens)
5 / 12THR A1033
ILE A 942
PHE A 901
PHE A 897
LEU A 895
None
1.40A16.43
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
1l9x GAMMA-GLUTAMYL
HYDROLASE
(Homo
sapiens)
5 / 12SER A 205
THR A 195
ILE A 204
LEU A 157
PHE A 113
None
1.36A24.07
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
1nd7 WW DOMAIN-CONTAINING
PROTEIN 1
(Homo
sapiens)
5 / 12SER A 580
TRP A 615
THR A 676
LEU A 592
PHE A 776
None
1.34A21.22
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
2osa N-CHIMAERIN
(Homo
sapiens)
5 / 12THR A 356
ILE A 352
LEU A 401
PHE A 347
LEU A 343
None
1.05A21.80
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3cxl N-CHIMERIN
(Homo
sapiens)
5 / 12THR A 356
ILE A 352
LEU A 401
PHE A 347
LEU A 343
None
1.12A20.55
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3pbl D(3) DOPAMINE
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
7 / 12THR A 115
ILE A 118
PHE A 338
TRP A 342
PHE A 345
PHE A 346
TYR A 373
None
None
None
None
ETQ  A1200 (-4.4A)
ETQ  A1200 ( 4.5A)
ETQ  A1200 (-4.4A)
0.54A30.47
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3pds FUSION PROTEIN
BETA-2 ADRENERGIC
RECEPTOR/LYSOZYME
(Homo
sapiens;
Escherichia
virus
T4)
8 / 12TRP A 109
THR A 118
ILE A 121
PHE A 282
TRP A 286
PHE A 289
PHE A 290
TYR A 316
None
None
None
None
None
ERC  A1201 (-4.5A)
ERC  A1201 (-4.8A)
None
0.69A30.32
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3rze HISTAMINE H1
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
8 / 12TRP A 103
SER A 111
THR A 112
ILE A 115
PHE A 424
TRP A 428
PHE A 432
TYR A 458
None
5EH  A1200 ( 3.7A)
D7V  A1201 ( 4.0A)
D7V  A1201 (-3.8A)
None
5EH  A1200 ( 3.4A)
5EH  A1200 ( 4.3A)
5EH  A1200 ( 4.4A)
0.53A28.10
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3u3z MICROCEPHALIN
(Homo
sapiens)
5 / 12SER A 819
THR A 821
ILE A 820
PHE A 756
LEU A 833
None
1.19A17.60
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4bqa PROTEIN C-ETS-2
(Homo
sapiens)
5 / 12LEU A 354
PHE A 442
PHE A 391
LEU A 446
TYR A 424
None
1.13A16.61
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4gbr BETA-2 ADRENERGIC
RECEPTOR
(Homo
sapiens)
8 / 12TRP A 109
THR A 118
ILE A 121
PHE A 254
TRP A 258
PHE A 261
PHE A 262
TYR A 288
None
CAU  A 500 ( 4.7A)
None
None
None
CAU  A 500 (-4.2A)
CAU  A 500 (-4.6A)
CAU  A 500 (-4.6A)
0.67A29.19
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4ib4 CHIMERA PROTEIN OF
HUMAN
5-HYDROXYTRYPTAMINE
RECEPTOR 2B AND E.
COLI SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
5 / 12LEU A 132
PHE A 333
TRP A 337
PHE A 341
TYR A 370
None
None
None
None
ERM  A2001 ( 4.8A)
1.41A62.50
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4ib4 CHIMERA PROTEIN OF
HUMAN
5-HYDROXYTRYPTAMINE
RECEPTOR 2B AND E.
COLI SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
7 / 12TRP A 131
SER A 139
THR A 140
ILE A 143
PHE A 340
PHE A 341
TYR A 370
None
ERM  A2001 (-3.6A)
ERM  A2001 (-3.9A)
None
ERM  A2001 (-4.3A)
None
ERM  A2001 ( 4.8A)
0.73A62.50
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4ib4 CHIMERA PROTEIN OF
HUMAN
5-HYDROXYTRYPTAMINE
RECEPTOR 2B AND E.
COLI SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
8 / 12TRP A 131
SER A 139
THR A 140
TRP A 337
PHE A 340
PHE A 341
LEU A 362
TYR A 370
None
ERM  A2001 (-3.6A)
ERM  A2001 (-3.9A)
None
ERM  A2001 (-4.3A)
None
ERM  A2001 ( 4.1A)
ERM  A2001 ( 4.8A)
0.76A62.50
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4ib4 CHIMERA PROTEIN OF
HUMAN
5-HYDROXYTRYPTAMINE
RECEPTOR 2B AND E.
COLI SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
7 / 12TRP A 131
THR A 140
ILE A 143
PHE A 333
PHE A 340
PHE A 341
TYR A 370
None
ERM  A2001 (-3.9A)
None
None
ERM  A2001 (-4.3A)
None
ERM  A2001 ( 4.8A)
0.90A62.50
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4ib4 CHIMERA PROTEIN OF
HUMAN
5-HYDROXYTRYPTAMINE
RECEPTOR 2B AND E.
COLI SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
8 / 12TRP A 131
THR A 140
PHE A 333
TRP A 337
PHE A 340
PHE A 341
LEU A 362
TYR A 370
None
ERM  A2001 (-3.9A)
None
None
ERM  A2001 (-4.3A)
None
ERM  A2001 ( 4.1A)
ERM  A2001 ( 4.8A)
0.86A62.50
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4lde LYSOZYME, BETA-2
ADRENERGIC RECEPTOR
(Homo
sapiens;
Escherichia
virus
T4)
6 / 12TRP A1109
THR A1118
ILE A1121
PHE A1289
PHE A1290
TYR A1316
None
None
None
P0G  A1401 ( 4.7A)
P0G  A1401 ( 4.9A)
None
0.87A24.22
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4lde LYSOZYME, BETA-2
ADRENERGIC RECEPTOR
(Homo
sapiens;
Escherichia
virus
T4)
6 / 12TRP A1109
THR A1118
TRP A1286
PHE A1289
PHE A1290
TYR A1316
None
None
None
P0G  A1401 ( 4.7A)
P0G  A1401 ( 4.9A)
None
0.68A24.22
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5i2x ADRENOCORTICAL
DYSPLASIA PROTEIN
HOMOLOG
(Homo
sapiens)
5 / 12SER A 165
THR A 164
TRP A 167
PHE A 173
LEU A 117
None
1.38A16.98
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5v54 5-HYDROXYTRYPTAMINE
RECEPTOR 1B,OB-1
FUSED 5-HT1B
RECEPTOR,5-HYDROXYTR
YPTAMINE RECEPTOR 1B
(Spodoptera
frugiperda;
Homo
sapiens)
8 / 12SER A 106
TRP A 125
THR A 134
ILE A 137
PHE A 323
TRP A 327
PHE A 330
PHE A 331
None
None
89F  A1201 (-4.2A)
None
None
89F  A1201 (-3.6A)
89F  A1201 (-4.1A)
89F  A1201 (-4.6A)
0.87Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5v54 5-HYDROXYTRYPTAMINE
RECEPTOR 1B,OB-1
FUSED 5-HT1B
RECEPTOR,5-HYDROXYTR
YPTAMINE RECEPTOR 1B
(Spodoptera
frugiperda;
Homo
sapiens)
8 / 12SER A 106
TRP A 125
THR A 134
ILE A 137
TRP A 327
PHE A 330
PHE A 331
TYR A 359
None
None
89F  A1201 (-4.2A)
None
89F  A1201 (-3.6A)
89F  A1201 (-4.1A)
89F  A1201 (-4.6A)
None
0.63Aundetectable
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5wiv D(4) DOPAMINE
RECEPTOR, SOLUBLE
CYTOCHROME B562
CHIMERA
(Escherichia
coli;
Homo
sapiens)
7 / 12THR A 120
ILE A 123
PHE A 403
TRP A 407
PHE A 410
PHE A 411
TYR A 438
AQD  A1201 (-4.4A)
None
None
None
AQD  A1201 (-4.7A)
AQD  A1201 (-4.6A)
None
0.78A44.91
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6bqh 5-HYDROXYTRYPTAMINE
RECEPTOR 2C,SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
11 / 12SER A 110
TRP A 130
SER A 138
THR A 139
ILE A 142
PHE A 320
TRP A 324
PHE A 327
PHE A 328
LEU A 350
TYR A 358
E2J  A1201 ( 4.5A)
None
E2J  A1201 (-3.2A)
E2J  A1201 (-4.3A)
E2J  A1201 (-3.5A)
E2J  A1201 (-4.4A)
E2J  A1201 ( 3.7A)
E2J  A1201 (-4.6A)
E2J  A1201 (-4.4A)
E2J  A1201 ( 4.3A)
None
0.49Aundetectable
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6cm4 D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
6 / 12THR A 119
PHE A 382
TRP A 386
PHE A 389
PHE A 390
TYR A 416
8NU  A2001 ( 4.4A)
8NU  A2001 ( 4.7A)
8NU  A2001 ( 3.8A)
8NU  A2001 ( 4.5A)
8NU  A2001 ( 4.8A)
8NU  A2001 ( 4.9A)
0.53A33.18
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6eua ANGIOPOIETIN-RELATED
PROTEIN 3
(Homo
sapiens)
5 / 12LEU A 362
PHE A 306
TRP A 314
PHE A 381
LEU A 351
None
1.32Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6g79 5-HYDROXYTRYPTAMINE
RECEPTOR 1B
(Homo
sapiens)
7 / 12SER S 106
TRP S 125
THR S 134
TRP S 327
PHE S 330
PHE S 331
TYR S 359
None
None
EP5  S 401 (-3.8A)
None
EP5  S 401 (-4.0A)
EP5  S 401 (-4.7A)
EP5  S 401 ( 4.9A)
0.81Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_A_8NUA3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6g79 5-HYDROXYTRYPTAMINE
RECEPTOR 1B
(Homo
sapiens)
5 / 12THR S 134
PHE S 323
TRP S 327
PHE S 330
PHE S 331
EP5  S 401 (-3.8A)
None
None
EP5  S 401 (-4.0A)
EP5  S 401 (-4.7A)
1.34Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
1ly7 FRATAXIN
(Homo
sapiens)
5 / 12THR A 191
PHE A 110
PHE A 109
LEU A 132
VAL A 134
None
1.06A16.27
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
1nd7 WW DOMAIN-CONTAINING
PROTEIN 1
(Homo
sapiens)
5 / 12SER A 580
TRP A 615
THR A 676
LEU A 592
PHE A 776
None
1.32A21.22
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
1o1u GASTROTROPIN
(Homo
sapiens)
5 / 12SER A  69
VAL A  91
THR A 100
PHE A  47
PHE A   2
None
1.14A13.16
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
1pcg ESTROGEN RECEPTOR
(Homo
sapiens)
6 / 12TYR A 328
VAL A 392
SER A 432
THR A 431
LEU A 349
LEU A 408
None
None
None
None
EST  A   1 ( 4.8A)
None
1.49A21.95
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
1szb MANNOSE BINDING
LECTIN-ASSOCIATED
SERINE PROTEASE-2
RELATED PROTEIN,
MAP19 (19KDA)
(Homo
sapiens)
5 / 12TYR A  92
THR A  82
LEU A  71
PHE A  49
LEU A  44
TYR  A  92 ( 1.3A)
THR  A  82 ( 0.8A)
LEU  A  71 ( 0.6A)
PHE  A  49 ( 1.3A)
LEU  A  44 ( 0.6A)
1.31A19.18
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
1wl4 ACETYL-COENZYME A
ACETYLTRANSFERASE 2
(Homo
sapiens)
5 / 12THR A 306
LEU A  96
TRP A 310
LEU A 366
VAL A 394
None
1.30A23.15
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
2a1r POLY(A)-SPECIFIC
RIBONUCLEASE PARN
(Homo
sapiens)
5 / 12TYR A  54
VAL A 284
LEU A 290
PHE A  69
VAL A 297
None
1.26A21.18
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
2b49 PROTEIN TYROSINE
PHOSPHATASE,
NON-RECEPTOR TYPE 3
(Homo
sapiens)
5 / 12VAL A 840
THR A 849
LEU A 831
PHE A 824
PHE A 821
None
1.36A19.47
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
2ckh SENTRIN-SPECIFIC
PROTEASE 1
(Homo
sapiens)
5 / 12VAL A 509
LEU A 567
PHE A 493
LEU A 524
VAL A 526
None
1.30A18.64
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3cem GLYCOGEN
PHOSPHORYLASE, LIVER
FORM
(Homo
sapiens)
5 / 12LEU A 581
PHE A 750
PHE A 749
LEU A 622
VAL A 626
None
1.31A18.79
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3o57 CAMP-SPECIFIC
3',5'-CYCLIC
PHOSPHODIESTERASE 4B
(Homo
sapiens)
5 / 12VAL A 371
THR A 367
LEU A 250
LEU A 384
VAL A 383
None
1.10A21.61
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3pbl D(3) DOPAMINE
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12VAL A 111
THR A 115
TRP A 342
PHE A 345
PHE A 346
ETQ  A1200 (-3.4A)
None
None
ETQ  A1200 (-4.4A)
ETQ  A1200 ( 4.5A)
0.44A30.47
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3pds FUSION PROTEIN
BETA-2 ADRENERGIC
RECEPTOR/LYSOZYME
(Homo
sapiens;
Escherichia
virus
T4)
6 / 12TRP A 109
VAL A 114
THR A 118
TRP A 286
PHE A 289
PHE A 290
None
ERC  A1201 (-3.8A)
None
None
ERC  A1201 (-4.5A)
ERC  A1201 (-4.8A)
0.51A30.32
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3rze HISTAMINE H1
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12TRP A 103
SER A 111
THR A 112
TRP A 428
PHE A 432
None
5EH  A1200 ( 3.7A)
D7V  A1201 ( 4.0A)
5EH  A1200 ( 3.4A)
5EH  A1200 ( 4.3A)
0.58A28.10
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3zrh UBIQUITIN
THIOESTERASE ZRANB1
(Homo
sapiens)
5 / 12VAL A 528
THR A 524
LEU A 375
LEU A 449
VAL A 448
None
1.29A22.97
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4asc KELCH REPEAT AND BTB
DOMAIN-CONTAINING
PROTEIN 5
(Homo
sapiens)
5 / 12VAL A 363
SER A 353
PHE A 321
LEU A 613
VAL A 611
None
1.14A23.21
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4bkf EPHRIN-B3
(Homo
sapiens)
5 / 12TYR C  51
LEU C  30
TRP C  35
LEU C 165
VAL C 163
None
1.18A17.77
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4fww MACROPHAGE-STIMULATI
NG PROTEIN RECEPTOR
(Homo
sapiens)
5 / 12VAL A 461
THR A 454
LEU A 483
LEU A 443
VAL A 366
None
1.27A21.03
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4gbr BETA-2 ADRENERGIC
RECEPTOR
(Homo
sapiens)
6 / 12TRP A 109
VAL A 114
THR A 118
TRP A 258
PHE A 261
PHE A 262
None
CAU  A 500 (-3.5A)
CAU  A 500 ( 4.7A)
None
CAU  A 500 (-4.2A)
CAU  A 500 (-4.6A)
0.51A29.19
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4ib4 CHIMERA PROTEIN OF
HUMAN
5-HYDROXYTRYPTAMINE
RECEPTOR 2B AND E.
COLI SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
7 / 12TRP A 131
VAL A 136
SER A 139
THR A 140
PHE A 340
PHE A 341
VAL A 366
None
ERM  A2001 (-3.8A)
ERM  A2001 (-3.6A)
ERM  A2001 (-3.9A)
ERM  A2001 (-4.3A)
None
ERM  A2001 ( 4.2A)
0.73A62.50
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4ib4 CHIMERA PROTEIN OF
HUMAN
5-HYDROXYTRYPTAMINE
RECEPTOR 2B AND E.
COLI SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
8 / 12TRP A 131
VAL A 136
SER A 139
TRP A 337
PHE A 340
PHE A 341
LEU A 362
VAL A 366
None
ERM  A2001 (-3.8A)
ERM  A2001 (-3.6A)
None
ERM  A2001 (-4.3A)
None
ERM  A2001 ( 4.1A)
ERM  A2001 ( 4.2A)
0.82A62.50
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4lde LYSOZYME, BETA-2
ADRENERGIC RECEPTOR
(Homo
sapiens;
Escherichia
virus
T4)
6 / 12TRP A1109
VAL A1114
THR A1118
TRP A1286
PHE A1289
PHE A1290
None
P0G  A1401 (-3.7A)
None
None
P0G  A1401 ( 4.7A)
P0G  A1401 ( 4.9A)
0.70A24.22
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4qt8 MACROPHAGE-STIMULATI
NG PROTEIN RECEPTOR
(Homo
sapiens)
5 / 12VAL B 461
THR B 454
LEU B 483
LEU B 443
VAL B 366
None
1.31A20.12
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5i2x ADRENOCORTICAL
DYSPLASIA PROTEIN
HOMOLOG
(Homo
sapiens)
5 / 12SER A 165
THR A 164
TRP A 167
PHE A 173
LEU A 117
None
1.37A16.98
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5neu INTEGRIN ALPHA-V
(Homo
sapiens)
5 / 12SER A 225
SER A 316
THR A 329
PHE A 267
VAL A 253
None
0.99A21.10
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5v54 5-HYDROXYTRYPTAMINE
RECEPTOR 1B,OB-1
FUSED 5-HT1B
RECEPTOR,5-HYDROXYTR
YPTAMINE RECEPTOR 1B
(Spodoptera
frugiperda;
Homo
sapiens)
6 / 12SER A 106
TRP A 125
THR A 134
TRP A 327
PHE A 330
PHE A 331
None
None
89F  A1201 (-4.2A)
89F  A1201 (-3.6A)
89F  A1201 (-4.1A)
89F  A1201 (-4.6A)
0.53Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5w0m TERMINAL
URIDYLYLTRANSFERASE
7
(Homo
sapiens)
5 / 12SER A1233
VAL A1004
LEU A1239
PHE A 997
LEU A 993
None
1.35A22.20
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5w0m TERMINAL
URIDYLYLTRANSFERASE
7
(Homo
sapiens)
5 / 12SER A1233
VAL A1004
LEU A1239
PHE A1318
LEU A 993
None
1.29A22.20
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5wiv D(4) DOPAMINE
RECEPTOR, SOLUBLE
CYTOCHROME B562
CHIMERA
(Escherichia
coli;
Homo
sapiens)
5 / 12VAL A 116
THR A 120
TRP A 407
PHE A 410
PHE A 411
AQD  A1201 ( 3.9A)
AQD  A1201 (-4.4A)
None
AQD  A1201 (-4.7A)
AQD  A1201 (-4.6A)
0.72A44.91
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6bqh 5-HYDROXYTRYPTAMINE
RECEPTOR 2C,SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
10 / 12SER A 110
TRP A 130
VAL A 135
SER A 138
THR A 139
TRP A 324
PHE A 327
PHE A 328
LEU A 350
VAL A 354
E2J  A1201 ( 4.5A)
None
E2J  A1201 (-3.8A)
E2J  A1201 (-3.2A)
E2J  A1201 (-4.3A)
E2J  A1201 ( 3.7A)
E2J  A1201 (-4.6A)
E2J  A1201 (-4.4A)
E2J  A1201 ( 4.3A)
E2J  A1201 (-4.6A)
0.58Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6bqh 5-HYDROXYTRYPTAMINE
RECEPTOR 2C,SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
10 / 12SER A 110
TYR A 118
TRP A 130
VAL A 135
THR A 139
TRP A 324
PHE A 327
PHE A 328
LEU A 350
VAL A 354
E2J  A1201 ( 4.5A)
None
None
E2J  A1201 (-3.8A)
E2J  A1201 (-4.3A)
E2J  A1201 ( 3.7A)
E2J  A1201 (-4.6A)
E2J  A1201 (-4.4A)
E2J  A1201 ( 4.3A)
E2J  A1201 (-4.6A)
0.68Aundetectable
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6cm4 D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12VAL A 115
THR A 119
TRP A 386
PHE A 389
PHE A 390
8NU  A2001 ( 3.5A)
8NU  A2001 ( 4.4A)
8NU  A2001 ( 3.8A)
8NU  A2001 ( 4.5A)
8NU  A2001 ( 4.8A)
0.45A33.18
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6g79 5-HYDROXYTRYPTAMINE
RECEPTOR 1B
(Homo
sapiens)
5 / 12SER S 106
TRP S 125
THR S 134
PHE S 330
PHE S 331
None
None
EP5  S 401 (-3.8A)
EP5  S 401 (-4.0A)
EP5  S 401 (-4.7A)
0.79Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_0
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6g79 5-HYDROXYTRYPTAMINE
RECEPTOR 1B
(Homo
sapiens)
5 / 12SER S 106
TRP S 125
TRP S 327
PHE S 330
PHE S 331
None
None
None
EP5  S 401 (-4.0A)
EP5  S 401 (-4.7A)
0.72Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
1yck PEPTIDOGLYCAN
RECOGNITION PROTEIN
(Homo
sapiens)
4 / 5ASP A  81
ILE A 124
ASN A  58
TYR A  85
None
0.98A18.78
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3pbl D(3) DOPAMINE
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
4 / 5ASP A 110
ILE A 118
PHE A 338
TYR A 373
ETQ  A1200 (-3.5A)
None
None
ETQ  A1200 (-4.4A)
0.46A30.47
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3pds FUSION PROTEIN
BETA-2 ADRENERGIC
RECEPTOR/LYSOZYME
(Homo
sapiens;
Escherichia
virus
T4)
4 / 5ASP A 113
ILE A 121
PHE A 282
TYR A 316
ERC  A1201 (-3.7A)
None
None
None
0.64A30.32
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3rze HISTAMINE H1
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
4 / 5ASP A 107
ILE A 115
PHE A 424
TYR A 458
5EH  A1200 ( 2.6A)
D7V  A1201 (-3.8A)
None
5EH  A1200 ( 4.4A)
0.48A28.10
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3she MAP KINASE-ACTIVATED
PROTEIN KINASE 3
(Homo
sapiens)
4 / 5ASP A 149
ILE A 130
PHE A 138
ASN A 305
None
1.21A21.13
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3u2p RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-4
(Homo
sapiens)
4 / 5ILE A 379
PHE A 389
ASN A 470
TYR A 444
None
None
NAG  A1005 (-1.8A)
None
1.10A21.66
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
3u7u RECEPTOR
TYROSINE-PROTEIN
KINASE ERBB-4
(Homo
sapiens)
4 / 5ILE A 379
PHE A 389
ASN A 470
TYR A 444
None
1.25A19.36
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4gbr BETA-2 ADRENERGIC
RECEPTOR
(Homo
sapiens)
4 / 5ASP A 113
ILE A 121
PHE A 254
TYR A 288
CAU  A 500 (-3.0A)
None
None
CAU  A 500 (-4.6A)
0.59A29.19
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4h1s 5'-NUCLEOTIDASE
(Homo
sapiens)
4 / 5ASP A 226
ILE A  31
ASN A 117
TYR A 176
None
None
ZN  A 602 ( 2.7A)
None
1.19A21.15
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4owt INTEGRATOR COMPLEX
SUBUNIT 3
(Homo
sapiens)
4 / 5ASP A 117
ILE A 126
PHE A  94
ASN A  76
None
1.20A22.29
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4rwa SOLUBLE CYTOCHROME
B562,DELTA-TYPE
OPIOID RECEPTOR
(Escherichia
coli;
Homo
sapiens)
4 / 5ASP A 128
ILE A 136
PHE A 270
TYR A 308
None
0.58A21.71
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
4zdv MICROTUBULE-ASSOCIAT
ED PROTEINS 1A/1B
LIGHT CHAIN 3A
(Homo
sapiens)
4 / 5ASP A 106
ILE A  23
ASN A  84
TYR A 110
None
0.93A16.12
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5clw 1,4-ALPHA-GLUCAN-BRA
NCHING ENZYME
(Homo
sapiens)
4 / 5ASP A 286
ILE A 206
PHE A 551
TYR A 251
None
1.08A20.44
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5dst PROTEIN ARGININE
N-METHYLTRANSFERASE
8
(Homo
sapiens)
4 / 5ASP A  92
ILE A 124
PHE A 128
ASN A 312
None
1.18A21.27
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5lsk PROTEIN MIS12
HOMOLOG
POLYAMINE-MODULATED
FACTOR 1
(Homo
sapiens;
Homo
sapiens)
4 / 5ASP B  39
ILE B  88
PHE A  28
ASN B 100
None
1.24A16.80
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5wiv D(4) DOPAMINE
RECEPTOR, SOLUBLE
CYTOCHROME B562
CHIMERA
(Escherichia
coli;
Homo
sapiens)
4 / 5ASP A 115
ILE A 123
PHE A 403
TYR A 438
AQD  A1201 (-3.3A)
None
None
None
0.41A44.91
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
5x49 PROBABLE XAA-PRO
AMINOPEPTIDASE 3
(Homo
sapiens)
4 / 5ILE A 343
PHE A 266
ASN A 319
TYR A 283
None
1.15A20.29
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6bqh 5-HYDROXYTRYPTAMINE
RECEPTOR 2C,SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
5 / 5ASP A 134
ILE A 142
PHE A 320
ASN A 351
TYR A 358
E2J  A1201 (-3.0A)
E2J  A1201 (-3.5A)
E2J  A1201 (-4.4A)
E2J  A1201 (-3.8A)
None
0.47Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6A93_B_8NUB3001_1
(5-HYDROXYTRYPTAMINE
RECEPTOR 2A,SOLUBLE
CYTOCHROME B562)
6c0t CGMP-DEPENDENT
PROTEIN KINASE 1
(Homo
sapiens)
4 / 5ASP A 597
ILE A 591
PHE A 579
ASN A 568
None
1.03Aundetectable
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
3pbl D(3) DOPAMINE
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
8 / 12PHE A 106
VAL A 111
THR A 115
PHE A 338
TRP A 342
PHE A 346
THR A 369
TYR A 373
ETQ  A1200 (-4.8A)
ETQ  A1200 (-3.4A)
None
None
None
ETQ  A1200 ( 4.5A)
ETQ  A1200 (-4.5A)
ETQ  A1200 (-4.4A)
0.69A74.84
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
3pbl D(3) DOPAMINE
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12VAL A 111
CYH A 114
THR A 115
TRP A 342
THR A 369
ETQ  A1200 (-3.4A)
ETQ  A1200 (-4.0A)
None
None
ETQ  A1200 (-4.5A)
1.16A74.84
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
3pbl D(3) DOPAMINE
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12VAL A 111
CYH A 114
THR A 115
TRP A 342
TYR A 365
ETQ  A1200 (-3.4A)
ETQ  A1200 (-4.0A)
None
None
None
1.34A74.84
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
3pbl D(3) DOPAMINE
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12VAL A 111
SER A 192
PHE A 338
TRP A 342
PHE A 346
ETQ  A1200 (-3.4A)
ETQ  A1200 (-3.3A)
None
None
ETQ  A1200 ( 4.5A)
0.98A74.84
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
3pbl D(3) DOPAMINE
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
6 / 12VAL A 111
THR A 115
PHE A 338
TRP A 342
PHE A 346
TYR A 365
ETQ  A1200 (-3.4A)
None
None
None
ETQ  A1200 ( 4.5A)
None
0.90A74.84
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
3pds FUSION PROTEIN
BETA-2 ADRENERGIC
RECEPTOR/LYSOZYME
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12PHE A 282
TRP A 286
PHE A 290
TYR A 308
TYR A 316
None
None
ERC  A1201 (-4.8A)
None
None
0.84A57.61
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
3pds FUSION PROTEIN
BETA-2 ADRENERGIC
RECEPTOR/LYSOZYME
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12SER A 203
PHE A 282
TRP A 286
PHE A 290
TYR A 308
ERC  A1201 (-2.8A)
None
None
ERC  A1201 (-4.8A)
None
1.06A57.61
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
3pds FUSION PROTEIN
BETA-2 ADRENERGIC
RECEPTOR/LYSOZYME
(Homo
sapiens;
Escherichia
virus
T4)
6 / 12VAL A 114
THR A 118
PHE A 282
TRP A 286
PHE A 290
TYR A 316
ERC  A1201 (-3.8A)
None
None
None
ERC  A1201 (-4.8A)
None
0.73A57.61
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
3pds FUSION PROTEIN
BETA-2 ADRENERGIC
RECEPTOR/LYSOZYME
(Homo
sapiens;
Escherichia
virus
T4)
6 / 12VAL A 114
THR A 118
SER A 203
PHE A 282
TRP A 286
PHE A 290
ERC  A1201 (-3.8A)
None
ERC  A1201 (-2.8A)
None
None
ERC  A1201 (-4.8A)
0.92A57.61
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
3rze HISTAMINE H1
RECEPTOR, LYSOZYME
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12THR A 112
PHE A 424
TRP A 428
PHE A 432
TYR A 458
D7V  A1201 ( 4.0A)
None
5EH  A1200 ( 3.4A)
5EH  A1200 ( 4.3A)
5EH  A1200 ( 4.4A)
0.55A58.04
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
4gbr BETA-2 ADRENERGIC
RECEPTOR
(Homo
sapiens)
5 / 12PHE A 254
TRP A 258
PHE A 262
TYR A 280
TYR A 288
None
None
CAU  A 500 (-4.6A)
None
CAU  A 500 (-4.6A)
0.64A25.59
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
4gbr BETA-2 ADRENERGIC
RECEPTOR
(Homo
sapiens)
6 / 12VAL A 114
THR A 118
PHE A 254
TRP A 258
PHE A 262
TYR A 288
CAU  A 500 (-3.5A)
CAU  A 500 ( 4.7A)
None
None
CAU  A 500 (-4.6A)
CAU  A 500 (-4.6A)
0.74A25.59
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
4ib4 CHIMERA PROTEIN OF
HUMAN
5-HYDROXYTRYPTAMINE
RECEPTOR 2B AND E.
COLI SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
6 / 12VAL A 136
THR A 140
PHE A 333
TRP A 337
PHE A 341
TYR A 370
ERM  A2001 (-3.8A)
ERM  A2001 (-3.9A)
None
None
None
ERM  A2001 ( 4.8A)
1.03A30.04
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
4lde LYSOZYME, BETA-2
ADRENERGIC RECEPTOR
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12VAL A1114
THR A1118
SER A1203
TRP A1286
PHE A1290
P0G  A1401 (-3.7A)
None
P0G  A1401 (-2.9A)
None
P0G  A1401 ( 4.9A)
1.02A32.55
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
4lde LYSOZYME, BETA-2
ADRENERGIC RECEPTOR
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12VAL A1114
THR A1118
TRP A1286
PHE A1290
TYR A1316
P0G  A1401 (-3.7A)
None
None
P0G  A1401 ( 4.9A)
None
0.65A32.55
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
4m7f FIBRINOGEN C
DOMAIN-CONTAINING
PROTEIN 1
(Homo
sapiens)
5 / 12TRP A 410
PHE A 350
VAL A 333
SER A 450
TYR A 302
None
1.37A17.44
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
4r9j FICOLIN-2
(Homo
sapiens)
5 / 12TRP G 241
PHE G 185
VAL G 168
SER G 281
TYR G 137
None
1.42A19.67
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
5a31 ANAPHASE-PROMOTING
COMPLEX SUBUNIT 1
ANAPHASE-PROMOTING
COMPLEX SUBUNIT 2
(Homo
sapiens;
Homo
sapiens)
5 / 12VAL A1848
CYH A1850
THR A1851
PHE N 163
THR N 155
None
1.41A14.58
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
5v54 5-HYDROXYTRYPTAMINE
RECEPTOR 1B,OB-1
FUSED 5-HT1B
RECEPTOR,5-HYDROXYTR
YPTAMINE RECEPTOR 1B
(Spodoptera
frugiperda;
Homo
sapiens)
6 / 12CYH A 133
THR A 134
TRP A 327
PHE A 331
THR A 355
TYR A 359
89F  A1201 (-4.5A)
89F  A1201 (-4.2A)
89F  A1201 (-3.6A)
89F  A1201 (-4.6A)
89F  A1201 (-4.0A)
None
0.42Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
5v54 5-HYDROXYTRYPTAMINE
RECEPTOR 1B,OB-1
FUSED 5-HT1B
RECEPTOR,5-HYDROXYTR
YPTAMINE RECEPTOR 1B
(Spodoptera
frugiperda;
Homo
sapiens)
5 / 12THR A 134
PHE A 323
TRP A 327
PHE A 331
THR A 355
89F  A1201 (-4.2A)
None
89F  A1201 (-3.6A)
89F  A1201 (-4.6A)
89F  A1201 (-4.0A)
0.79Aundetectable
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
5wiv D(4) DOPAMINE
RECEPTOR, SOLUBLE
CYTOCHROME B562
CHIMERA
(Escherichia
coli;
Homo
sapiens)
5 / 12CYH A 119
THR A 120
SER A 197
TRP A 407
THR A 434
AQD  A1201 ( 3.9A)
AQD  A1201 (-4.4A)
AQD  A1201 ( 4.0A)
None
AQD  A1201 (-3.5A)
1.31A35.67
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
5wiv D(4) DOPAMINE
RECEPTOR, SOLUBLE
CYTOCHROME B562
CHIMERA
(Escherichia
coli;
Homo
sapiens)
5 / 12THR A 120
SER A 197
PHE A 403
TRP A 407
THR A 434
AQD  A1201 (-4.4A)
AQD  A1201 ( 4.0A)
None
None
AQD  A1201 (-3.5A)
1.00A35.67
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
5wiv D(4) DOPAMINE
RECEPTOR, SOLUBLE
CYTOCHROME B562
CHIMERA
(Escherichia
coli;
Homo
sapiens)
5 / 12VAL A 116
CYH A 119
THR A 120
TRP A 407
THR A 434
AQD  A1201 ( 3.9A)
AQD  A1201 ( 3.9A)
AQD  A1201 (-4.4A)
None
AQD  A1201 (-3.5A)
1.14A35.67
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
5wiv D(4) DOPAMINE
RECEPTOR, SOLUBLE
CYTOCHROME B562
CHIMERA
(Escherichia
coli;
Homo
sapiens)
6 / 12VAL A 116
PHE A 403
TRP A 407
PHE A 411
THR A 434
TYR A 438
AQD  A1201 ( 3.9A)
None
None
AQD  A1201 (-4.6A)
AQD  A1201 (-3.5A)
None
0.68A35.67
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
5wiv D(4) DOPAMINE
RECEPTOR, SOLUBLE
CYTOCHROME B562
CHIMERA
(Escherichia
coli;
Homo
sapiens)
5 / 12VAL A 116
SER A 196
PHE A 403
TRP A 407
PHE A 411
AQD  A1201 ( 3.9A)
AQD  A1201 (-2.8A)
None
None
AQD  A1201 (-4.6A)
1.12A35.67
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
5wiv D(4) DOPAMINE
RECEPTOR, SOLUBLE
CYTOCHROME B562
CHIMERA
(Escherichia
coli;
Homo
sapiens)
6 / 12VAL A 116
THR A 120
PHE A 403
TRP A 407
THR A 434
TYR A 438
AQD  A1201 ( 3.9A)
AQD  A1201 (-4.4A)
None
None
AQD  A1201 (-3.5A)
None
0.40A35.67
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
6bqh 5-HYDROXYTRYPTAMINE
RECEPTOR 2C,SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
5 / 12THR A 139
SER A 219
PHE A 320
TRP A 324
PHE A 328
E2J  A1201 (-4.3A)
E2J  A1201 (-3.2A)
E2J  A1201 (-4.4A)
E2J  A1201 ( 3.7A)
E2J  A1201 (-4.4A)
0.95Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
6bqh 5-HYDROXYTRYPTAMINE
RECEPTOR 2C,SOLUBLE
CYTOCHROME B562
(Escherichia
coli;
Homo
sapiens)
6 / 12VAL A 135
THR A 139
PHE A 320
TRP A 324
PHE A 328
TYR A 358
E2J  A1201 (-3.8A)
E2J  A1201 (-4.3A)
E2J  A1201 (-4.4A)
E2J  A1201 ( 3.7A)
E2J  A1201 (-4.4A)
None
0.40Aundetectable
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
6cm4 D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
5 / 12SER A 194
PHE A 382
TRP A 386
TYR A 408
THR A 412
None
8NU  A2001 ( 4.7A)
8NU  A2001 ( 3.8A)
8NU  A2001 ( 4.0A)
8NU  A2001 ( 3.8A)
0.79A100.00
Available target for annotated drug, i.e. matched protein structure has more than 30% sequence identity to known drug target.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
6cm4 D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
12 / 12TRP A 100
PHE A 110
VAL A 115
CYH A 118
THR A 119
SER A 193
PHE A 382
TRP A 386
PHE A 390
TYR A 408
THR A 412
TYR A 416
None
8NU  A2001 ( 4.9A)
8NU  A2001 ( 3.5A)
8NU  A2001 ( 4.0A)
8NU  A2001 ( 4.4A)
8NU  A2001 ( 4.5A)
8NU  A2001 ( 4.7A)
8NU  A2001 ( 3.8A)
8NU  A2001 ( 4.8A)
8NU  A2001 ( 4.0A)
8NU  A2001 ( 3.8A)
8NU  A2001 ( 4.9A)
0.00A100.00
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
6g79 5-HYDROXYTRYPTAMINE
RECEPTOR 1B
(Homo
sapiens)
5 / 12CYH S 133
THR S 134
PHE S 331
TYR S 109
TYR S 359
EP5  S 401 (-4.2A)
EP5  S 401 (-3.8A)
EP5  S 401 (-4.7A)
None
EP5  S 401 ( 4.9A)
1.34Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
6g79 5-HYDROXYTRYPTAMINE
RECEPTOR 1B
(Homo
sapiens)
5 / 12CYH S 133
THR S 134
TRP S 327
THR S 355
TYR S 359
EP5  S 401 (-4.2A)
EP5  S 401 (-3.8A)
None
None
EP5  S 401 ( 4.9A)
0.82Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_0
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
6g79 5-HYDROXYTRYPTAMINE
RECEPTOR 1B
(Homo
sapiens)
5 / 12CYH S 133
TRP S 327
PHE S 331
THR S 355
TYR S 359
EP5  S 401 (-4.2A)
None
EP5  S 401 (-4.7A)
None
EP5  S 401 ( 4.9A)
0.90Aundetectable
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_1
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
4zgz ANTIZYME INHIBITOR 1
ORNITHINE
DECARBOXYLASE
ANTIZYME 1
(Homo
sapiens;
Homo
sapiens)
4 / 4ASP A 387
ALA A  88
SER A  90
PHE B 192
None
1.41A22.99
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_1
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
5c5b DCC-INTERACTING
PROTEIN 13-ALPHA
(Homo
sapiens)
4 / 4ASP A  15
ALA A 142
SER A 170
PHE A 133
None
1.46A21.38
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_1
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
5xjy ATP-BINDING CASSETTE
SUB-FAMILY A MEMBER
1
(Homo
sapiens)
4 / 4ASP A1706
ALA A1766
SER A1757
PHE A1675
None
1.40A11.75
Potential target for repurposing, i.e. matched protein structure has less than 30% sequence identity to known drug target, and may potentially interact with the same drug molecule based on local structural similarity of binding site.
6CM4_A_8NUA2001_1
(D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA)
6cm4 D(2) DOPAMINE
RECEPTOR, ENDOLYSIN
CHIMERA
(Homo
sapiens;
Escherichia
virus
T4)
4 / 4ASP A 114
ALA A 122
SER A 197
PHE A 389
8NU  A2001 ( 3.0A)
8NU  A2001 ( 3.3A)
8NU  A2001 ( 3.6A)
8NU  A2001 ( 4.5A)
0.01Aundetectable