KNOWN TARGETS FROM HUMAN (PROTEIN-DRUG COMPLEXES IN THE PDB)

1) Click on the entry ID to view details of interfaces and pattern clusters
2) Note that ASSAM search use only 3-12 residue containing patterns
DrReposER ID PDB Ligand Organism Macromolecule Pfam Res. Interface HETATM View
3TVX_A_PNXA902 3tvx PNX

DB00806
(Pentoxifylline)
Homo sapiens CAMP-SPECIFIC
3',5'-CYCLIC
PHOSPHODIESTERASE 4A
PF00233
(PDEase_I)
9 TYR A 371
LEU A 531
ASN A 533
PRO A 534
THR A 545
ILE A 548
MET A 569
GLN A 581
PHE A 584
PNX A 902
3TVX_B_PNXB902 3tvx PNX

DB00806
(Pentoxifylline)
Homo sapiens CAMP-SPECIFIC
3',5'-CYCLIC
PHOSPHODIESTERASE 4A
no annotation 7 TYR B 371
ASN B 533
ILE B 548
PHE B 552
MET B 569
GLN B 581
PHE B 584
PNX B 902