KNOWN TARGETS FROM HUMAN (PROTEIN-DRUG COMPLEXES IN THE PDB)

1) Click on the entry ID to view details of interfaces and pattern clusters
2) Note that ASSAM search use only 3-12 residue containing patterns
DrReposER ID PDB Ligand Organism Macromolecule Pfam Res. Interface HETATM View
3HII_A_PNTA901 3hii PNT

DB00738
(Pentamidine)
Homo sapiens AMILORIDE-SENSITIVE
AMINE OXIDASE
None
PF01179
(Cu_amine_oxid)
PF02727
(Cu_amine_oxidN3)
PF02728
(Cu_amine_oxidN2)
13 TYR A 148
THR A 185
ASP A 186
TYR A 371
ASP A 373
TRP A 376
GLY A 377
SER A 380
VAL A 381
TYR A 404
PHE B 435
TYR A 459
ASN A 460
PNT A 901
3HII_B_PNTB901 3hii PNT

DB00738
(Pentamidine)
Homo sapiens AMILORIDE-SENSITIVE
AMINE OXIDASE
None 12 TYR B 148
THR B 185
ASP B 186
TYR B 371
ASP B 373
TRP B 376
GLY B 377
SER B 380
VAL B 381
TYR B 404
TYR B 459
ASN B 460
PNT B 901