KNOWN TARGETS FROM HUMAN (PROTEIN-DRUG COMPLEXES IN THE PDB)

1) Click on the entry ID to view details of interfaces and pattern clusters
2) Note that ASSAM search use only 3-12 residue containing patterns
DrReposER ID PDB Ligand Organism Macromolecule Pfam Res. Interface HETATM View
3W2T_A_LF7A801 3w2t LF7

DB04876
(Vildagliptin)
Homo sapiens DIPEPTIDYL PEPTIDASE
4
PF00326
(Peptidase_S9)
PF00930
(DPPIV_N)
12 ARG A 125
GLU A 205
GLU A 206
TYR A 547
SER A 630
TYR A 631
VAL A 656
TYR A 662
TYR A 666
ASN A 710
VAL A 711
HIS A 740
LF7 A 801
3W2T_B_LF7B801 3w2t LF7

DB04876
(Vildagliptin)
Homo sapiens DIPEPTIDYL PEPTIDASE
4
no annotation 12 ARG B 125
GLU B 205
GLU B 206
TYR B 547
SER B 630
TYR B 631
VAL B 656
TYR B 662
TYR B 666
ASN B 710
VAL B 711
HIS B 740
LF7 B 801
6B1E_A_LF7A801 6b1e LF7

DB04876
(Vildagliptin)
Homo sapiens DIPEPTIDYL PEPTIDASE
4
PF00326
(Peptidase_S9)
PF00930
(DPPIV_N)
11 ARG A 125
GLU A 205
GLU A 206
TYR A 547
SER A 630
TYR A 631
VAL A 656
TYR A 662
TYR A 666
ASN A 710
VAL A 711
LF7 A 801
6B1E_B_LF7B801 6b1e LF7

DB04876
(Vildagliptin)
Homo sapiens DIPEPTIDYL PEPTIDASE
4
no annotation 12 ARG B 125
GLU B 205
GLU B 206
TYR B 547
SER B 630
TYR B 631
VAL B 656
TYR B 662
TYR B 666
ASN B 710
VAL B 711
HIS B 740
LF7 B 801