KNOWN TARGETS FROM HUMAN (PROTEIN-DRUG COMPLEXES IN THE PDB)

1) Click on the entry ID to view details of interfaces and pattern clusters
2) Note that ASSAM search use only 3-12 residue containing patterns
DrReposER ID PDB Ligand Organism Macromolecule Pfam Res. Interface HETATM View
1AVN_A_HSMA264 1avn HSM

DB05381
(Histamine)
Homo sapiens CARBONIC ANHYDRASE
II
PF00194
(Carb_anhydrase)
4 ASN A  62
HIS A  64
ASN A  67
GLN A  92
HSM A 264
1JQD_A_HSMA600 1jqd HSM

DB05381
(Histamine)
Homo sapiens HISTAMINE
N-METHYLTRANSFERASE
PF13489
(Methyltransf_23)
7 PHE A  22
GLU A  28
GLN A 143
VAL A 173
TRP A 179
TRP A 183
ASN A 283
HSM A 600
1JQD_B_HSMB601 1jqd HSM

DB05381
(Histamine)
Homo sapiens HISTAMINE
N-METHYLTRANSFERASE
no annotation 10 PHE B  22
GLU B  28
GLN B 143
TYR B 146
VAL B 173
TRP B 179
TRP B 183
PHE B 243
ASN B 283
LEU B 285
HSM B 601