KNOWN TARGETS FROM HUMAN (PROTEIN-DRUG COMPLEXES IN THE PDB)

1) Click on the entry ID to view details of interfaces and pattern clusters
2) Note that ASSAM search use only 3-12 residue containing patterns
DrReposER ID PDB Ligand Organism Macromolecule Pfam Res. Interface HETATM View
4HVC_A_HFGA1602 4hvc HFG

DB04866
(Halofuginone)
Homo sapiens BIFUNCTIONAL
GLUTAMATE/PROLINE--T
RNA LIGASE
PF00587
(HGTP_anticodon)
PF03129
(ProRS-C_1)
PF09180
(tRNA-synt_2b)
16 HIS A1093
PHE A1097
GLU A1100
VAL A1101
PRO A1120
THR A1121
GLU A1123
ARG A1152
TRP A1169
GLU A1171
HIS A1173
PHE A1216
THR A1240
HIS A1242
SER A1272
GLY A1274
HFG A1602
4HVC_B_HFGB1602 4hvc HFG

DB04866
(Halofuginone)
Homo sapiens BIFUNCTIONAL
GLUTAMATE/PROLINE--T
RNA LIGASE
None 17 LEU B1087
HIS B1093
PHE B1097
GLU B1100
VAL B1101
PRO B1120
THR B1121
GLU B1123
ARG B1152
TRP B1169
GLU B1171
HIS B1173
PHE B1216
THR B1240
HIS B1242
SER B1272
GLY B1274
HFG B1602
4K88_A_HFGA602 4k88 HFG

DB04866
(Halofuginone)
Homo sapiens PROLINE--TRNA LIGASE PF00587
(ProRS-C_1)
PF03129
(tRNA-synt_2b)
PF09180
(HGTP_anticodon)
12 PHE A  97
GLU A 100
VAL A 101
PRO A 120
THR A 121
GLU A 123
ARG A 152
TRP A 169
GLU A 171
PHE A 216
HIS A 242
SER A 272
HFG A 602