KNOWN TARGETS FROM HUMAN (PROTEIN-DRUG COMPLEXES IN THE PDB)

1) Click on the entry ID to view details of interfaces and pattern clusters
2) Note that ASSAM search use only 3-12 residue containing patterns
DrReposER ID PDB Ligand Organism Macromolecule Pfam Res. Interface HETATM View
1MCB_P_DHIP3 1mcb DHI

DB00117
(L-
Histidine)
;
Homo sapiens
IMMUNOGLOBULIN
LAMBDA DIMER MCG
(LIGHT CHAIN);
PEPTIDE
N-ACETYL-L-GLN-D-PHE
-L-HIS-D-PRO-OH
None
PF07654
(C1-set)
PF07686
(V-set)
5 GLN P   1
TYR A  34
TYR A  51
GLU A  52
TYR B  93
DHI P   3
1MCL_P_DHIP1 1mcl DHI

DB00117
(L-
Histidine)
;
Homo sapiens
IMMUNOGLOBULIN
LAMBDA DIMER MCG
(LIGHT CHAIN);
N-ACETYL-D-HIS-L-PRO
-OH
None
PF07654
(V-set)
PF07686
(C1-set)
5 PRO P   2
TYR A  51
GLU A  52
TYR B  93
PHE A  99
DHI P   1
1MCN_P_DHIP1 1mcn DHI

DB00117
(L-
Histidine)
;
Homo sapiens
IMMUNOGLOBULIN
LAMBDA DIMER MCG
(LIGHT CHAIN);
PEPTIDE
N-ACETYL-D-HIS-L-PRO
-NH2
None
PF07654
(V-set)
PF07686
(C1-set)
3 PRO P   2
TYR B  34
PHE A  99
DHI P   1
2EZ7_A_DHIA301 2ez7 DHI

DB00117
(L-
Histidine)
Homo sapiens CARBONIC ANHYDRASE 2 PF00194
(Carb_anhydrase)
6 TRP A   5
HIS A  64
ASN A  67
GLN A  92
THR A 200
PRO A 202
DHI A 301
2M2O_B_DHIB24 2m2o DHI

DB00117
(L-
Histidine)
Homo sapiens INSULIN B CHAIN PF00049
(Insulin)
6 ARG B  22
GLY B  23
PHE B  25
PRO B  28
LYS B  29
THR B  30
DHI B  24
2M2P_B_DHIB24 2m2p DHI

DB00117
(L-
Histidine)
Homo sapiens INSULIN B CHAIN PF00049
(Insulin)
3 TYR B  16
GLY B  23
PHE B  25
DHI B  24
6BEO_A_DHIA4 6beo DHI

DB00117
(L-
Histidine)
Homo sapiens (DPR)PY(DHI)PKDL(DGN
)
None 3 TYR A   3
PRO A   5
LEU A   8
DHI A   4